Stereoselective hydrofluorination of ynamides: a straightforward synthesis of novel α-fluoroenamides.

نویسندگان

  • Guillaume Compain
  • Kevin Jouvin
  • Agnès Martin-Mingot
  • Gwilherm Evano
  • Jérome Marrot
  • Sébastien Thibaudeau
چکیده

α-Fluoroenamides, potent rigid fluorinated bioisosters of ureas, have been synthesized by a highly regio- and stereo-selective hydrofluorination of ynamides in anhydrous HF. This reaction provides the first general entry to α-fluoroenamides and can easily be applied to a wide range of substrates.

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عنوان ژورنال:
  • Chemical communications

دوره 48 42  شماره 

صفحات  -

تاریخ انتشار 2012